Apixaban (Kev lag luam)
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Apixaban (Kev lag luam)

Apixaban (Kev lag luam)

CAS: 503612-47-3
Purity: 99% min
MF: C25H25N5O4
Muaj peev xwm: 200kg / M
Therapy Cheeb Tsam: Cardiovascular
VQ cov ntaub ntawv & kev tshuaj xyuas qhov chaw: Muaj

Hauj lwm lawm

Apixaban yog ib qho tshuaj anticoagulant siv los txo txoj kev pheej hmoo ntawm mob stroke thiab kab mob embolism hauv cov neeg mob uas tsis muaj valcular atrial fibrillation..
Ib qho tseem ceeb hauv kev pab peb cov neeg siv khoom ua ntej rau kev ua lag luam yog cov khoom lag luam teb. Peb ua tiav qhov no los ntawm kev ua kom tag nrho peb cov chaw ua haujlwm tau zoo thiab ua raws li cov qauv tshiab ntawm kev ua tau zoo, kev nyab xeeb, thiab kev tsim khoom. Kev sib cuam tshuam zoo ntawm kev lag luam thiab cov chaw tsim khoom tso cai rau cov tshuaj tiv thaiv sai rau kev hloov pauv hauv kev lag luam, kom peb tuaj yeem tiv thaiv kev tsis txaus thiab ua tau raws li qhov xav tau tam sim ntawd.
Apixaban yog ib qho kev xaiv inhibitor ntawm FXa. Nws tsis xav tau antithrombin III rau kev ua haujlwm antithrombotic. Apixaban inhibits dawb thiab clot-bound FXa, thiab kev ua haujlwm prothrombinase. Apixaban tsis muaj kev cuam tshuam ncaj qha rau platelet aggregation, tab sis tsis ncaj qha inhibits platelet aggregation induced los ntawm thrombin. Los ntawm inhibiting FXa, apixaban txo thrombin tiam thiab thrombus kev loj hlob.

 

1-(4-Methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]{{7} },5,6,7-tetrahydro-1H-pyrazolo[3,{14}}c]pyridine-3-carboxylic acid ethyl ester 503614-91-3 Apixaban nruab nrab
Acetic acid, 2-chloro-2-[2-(4-methoxyphenyl)hydrazinylidene], ethyl ester 27143-07-3 Apixaban nruab nrab
2(1H)-pyridine, 3-chloro-5, 6-dihydro-1-(4-}nitrophenyl) 536760-29-9 Apixaban nruab nrab
3-Morpholin-4-yl-1-[4-(2-oxopiperidin-1-yl)phenyl]-5,6- dihydro-1H-pyridin{10}}ib 545445-44-1 Apixaban nruab nrab
3-(4-Morpholinyl)-1-(4-nitrophenyl)-5, 6-dihydro-2(1H)-pyridinone 503615-03-0 Apixaban nruab nrab
Ethyl 1-(4-methoxyphenyl)-6-(4-nitrophenyl)-7-oxo-4,5,6,7-tetrahydro{ {9}}H-pyrazolo[3,{12}}c]pyridine-3 536759-91-8 Apixaban nruab nrab
ethyl 6-(4-aMinophenyl)-1-(4-Methoxyphenyl)-7-oxo-4,5,6,7-tetrahydro{ {9}}H-pyrazolo[3,4-c]pyridine-3-carboxylate 503615-07-4 Apixaban nruab nrab
1-(4-AMinophenyl)-5, 6-dihydro-3-(4-Morpholinyl)-2(1h)-pyridinone 1267610-26-3 Apixaban nruab nrab

 

Paub ntau ntxiv, thov koj xav tiv tauj​​sales02@pharmachemm.com (Neeg Ada Li).

 

Txais tos tuaj xyuas peb ntawm

CPHI Europe 2024Lub rooj muag zaub 1A 138-7Kaum Hli Ntuj 8-10 Milan ltalis
Pharmtech & Cov khoom xyaw 2024Booth CCC-76Nov 19-22 Moscow Russia.

 

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