
Aprocitentan hmoov
CAS: 1103522-45-7
MF: C16H14Br2N6O4S
MW: 546.19
Lub neej txee: 2 xyoos
Qhov zoo:
Qauv yog Muaj
Qhov zoo tshaj plaws thiab tus nqi zoo tshaj
COA, HPLC, MSDS muaj
Daim ntawv pov thawj: ISO, CTC, SGS, CQC
Qhov chaw ntawm Keeb Kwm: Shandong, Suav
Hauj lwm lawm
Ntau tus phooj ywg uas muaj ntshav siab paub txog kev mob ntshav siab thiab paub siv cov tshuaj tiv thaiv hypertensive, tab sis lawv cov ntshav siab tsis tuaj yeem poob, thiab 3-4 hom ntshav siab siv tsis tau. Qhov no yog refractory hypertension, yuav muaj kev daws teeb meem yav tom ntej, cov tshuaj ntshav siab tshiab yuav pab tau koj daws qhov teeb meem, cov tshuaj no tsis yog sartan, tsis yog PriApril, tsis yog dipine, tab sis cov tshuaj ntshav siab tshiab.
Thaum Lub Peb Hlis 20, 2024, FDA tau pom zoo cov tshuaj tshiab Aprocitentan rau kev kho mob ntshav siab refractory. Peb caug xyoo dhau los, thawj sartan antihypertensive tshuaj losartan tuaj nyob rau hauv kev ua lag luam, thiab txij thaum ntawd los, cov tshuaj antihypertensive tshiab tau tshwm sim, tab sis lawv yog tag nrho cov tswv cuab tshiab ntawm tsev neeg, thiab tsis muaj hom tshuaj antihypertensive tshiab tau tuaj rau hauv khw. Nws tuaj yeem hais tias Aprocitentan Powder yog thawj cov tshuaj ntshav siab tshiab hauv 30 xyoo.
Aprocitentan Powder yog ib qho endothelin receptor antagonist uas antagonizes endothelin receptors thiab tseem tuaj yeem txo cov paj hlwb kev xav thiab txo qis kev tso tawm ntawm aldosterone. Nws tsis tsuas yog txo cov ntshav siab, tab sis kuj tiv thaiv intima ntawm cov hlab ntsha thiab txo qhov tshwm sim ntawm arteriosclerosis. Txoj kev tshawb nrhiav pom tias Aprocitentan, raws li kev siv lwm cov tshuaj tiv thaiv kab mob siab, tuaj yeem txo cov ntshav siab ntxiv los ntawm 15mmHg, uas yog 6mmHg ntau dua li ntawm pawg tswj hwm qhov nruab nrab, thiab cov txiaj ntsig tseem ceeb heev. Yog li ntawd, kev kho mob ntawm refractory hypertension, ntsev-sensitive hypertension, lub raum kub siab, ntshav qab zib ua ke nrog kub siab kuj zoo dua, thiab cov nyhuv ntawm kev txo cov zis protein kuj zoo dua.
Cov kev mob tshwm sim tseem ceeb yog me me edema, tab sis tsis loj, tsis nce ntshav poov tshuaj, yog li nws muaj kev nyab xeeb.
| Melting point | 139-141 degree |
| Boiling point | 705.0± 70.0 degree (Tshaj tawm) |
| ceev | 1.841 ± 0.06 g / cm3 (Tswj) |
| cia temp. | -20 degree lub freezer |
| solubility | Chloroform (me ntsis, rhaub), Methanol (me ntsis, rhaub) |
| daim ntawv | Khoom |
| pka ua | 13.56 ± 0.60 (Tshaj tawm) |
| xim | Dawb rau Off-White |
ZOO TSHAJ PLAWS PARTNER- Jinan Jianfeng Tshuaj
Jianfeng Chemical yog lub tuam txhab kev tshawb fawb-tsav tshuaj.Peb muaj ntau tshaj 10 xyoo kev paub hauv lub tsev muag tshuaj. Feem ntau tsim cov tshuaj APIs, Pharmaceutical intermediate thiab cov khoom siv tshuaj pleev ib ce. Raws li cov khoom zoo thiab cov nqi sib tw, peb muaj lub koob npe nrov hauv Tuam Tshoj cov chaw muag tshuaj.
Nyob rau hauv lub hauv paus ntsiab lus ntawm "Quality Oriented", Jianfeng tau dhau daim ntawv pov thawj ntawm ISO9001: 2008 Kev Tswj Xyuas Zoo.

Yuav koom tes nrog peb li cas?
--Cia peb cov lus hais txog cov khoom koj xav tau.
--Kev piav qhia ntawm kev txiav txim kom muaj nuj nqis.
--Thov qhia rau peb paub koj qhov chaw nyob shipping.
--Tus thawj tswj kev muag khoom muab nqe lus rau koj thiab xa daim ntawv cog lus rau koj.
--Kev xa khoom tib hnub tom qab them nyiaj.


Cim npe nrov: aprocitentan hmoov, Tuam Tshoj, lwm tus neeg, manufacturers, hoobkas, lag luam wholesale, yuav, tej, nqe, kev muag, hauv Tshuag
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